5-hydroxymethyl Tolterodine (formate)
如果您对该产品感兴趣的话,可以
产品名称:
5-hydroxymethyl Tolterodine (formate)
产品型号:
GOY-Y0386
产品展商:
谷研
产品文档:
无相关文档
发布时间:2023-04-10
简单介绍
5-hydroxymethyl Tolterodine (formate)DMSO: soluble,Methanol: soluble
5-hydroxymethyl Tolterodine (formate)
的详细介绍
|
性能参数
|
|
产品名称
|
5-hydroxymethyl Tolterodine (formate)
|
|
规格
|
1mg
|
|
货号
|
GOY-Y0386
|
|
含量
|
>98.00%
|
|
CAS
|
380636-49-7
|
|
别名
|
N/A
|
|
|
|
化学名
|
N/A
|
分子式
|
C22H31NO2?CH2O2
|
|
分子量
|
分子 387.5
|
溶解度
|
DMSO: soluble,Methanol: soluble
|
|
储存条件
|
Store at -20°C
|
General tips
|
|
|
用途
|
仅供科研
|
价格
|
电询
|
|
|
|
详细内容
|
5-hydroxymethyl Tolterodine is an active metabolite of the muscarinic acetylcholine receptor antagonists tolterodine and fesoterodine . It is formed from tolterodine by the cytochrome P450 (CYP) isoform CYP2D6 and from fesoterodine by plasma esterases. 5-hydroxymethyl Tolterodine inhibits M1-5 muscarinic receptors with Ki values of 2.3, 2, 2.5, 2.8, and 2.9 nM, respectively, for the human receptors expressed in CHO cells. It selectively inhibits acetylcholine-induced bladder contraction over electrically induced salivation in anesthetized cats (ID50s = 15 and 40 nmol/kg, respectively).
|
公司正在销售的产品：
|
3,7-O-二咖啡?？?规格： HPLC≥98%;20mg
3,6-O-二咖啡?？?规格： HPLC≥98%;20mg
丹叶大黄素 规格： HPLC≥98%;20mg
冬绿苷 规格： HPLC≥98%;20mg
地黄苷D 规格： HPLC≥98%;5mg
地黄苷A 规格： HPLC≥98%;5mg
|
2-溴-6-甲氧基吡啶2-Bromo-6-methoxypyridine,97%40473-07-25ML
2-氯-6-甲氧基吡啶2-Chloro-6-methoxypyridine,98%17228-64-75G
4-苯基吡啶4-Phenylpyridine,97%939-23-15G
3-苯基吡啶3-Phenylpyridine,98%1008-88-45G
2-苯基吡啶2-Phenylpyridine,98%1008-89-55G
2-羟基-5-甲基吡啶2-Hydroxy-5-methylpyridine,97%1003-68-51G
|