Amastatin (hydrochloride)
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产品名称:
Amastatin (hydrochloride)
产品型号:
GOY-Y0554
产品展商:
谷研
产品文档:
无相关文档
发布时间:2023-04-11
简单介绍
Amastatin (hydrochloride)DMF: 10 mg/ml,DMSO: 2 mg/ml,Ethanol: 1 mg/ml,PBS (pH 7.2): 5 mg/ml
Amastatin (hydrochloride)
的详细介绍
性能参数
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产品名称
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Amastatin (hydrochloride)
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规格
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500μg 1mg 5mg 10mg
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货号
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GOY-Y0554
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含量
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>95.00%
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CAS
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100938-10-1
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别名
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N/A
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化学名
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N/A
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分子式
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C21H38N4O8?HCl
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分子量
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分子 511
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溶解度
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DMF: 10 mg/ml,DMSO: 2 mg/ml,Ethanol: 1 mg/ml,PBS (pH 7.2): 5 mg/ml
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储存条件
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Store at -20°C
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General tips
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用途
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仅供科研
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价格
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电询
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详细内容
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Amastatin is a slow, tight binding, competitive aminopeptidase (AP) inhibitor, first described as an inhibitor of human serum AP-A (glutamyl AP; IC50 = 0.54 μg/ml) but not of AP-B (arginine AP). It also inhibits AP-N (AP-M, alanyl AP; Ki = 20-200 nM), leucyl-cystinyl AP (Ki = 20-220 nM), and endoplasmic reticulum AP 1 (Ki = 41.8 μM). Amastatin is without effect on trypsin, papain, chymotrypsin, elastase, pepsin, or thermolysin.
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